PD153035
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


PD153035
Target:
EGFRRelated Pathways:
Angiogenesis|||JAK/STAT signaling|||Tyrosine Kinase/AdaptorsPurity:
0.9931Bioactivity:
PD153035 (NSC-669364) hydrochloride is an effective and selective inhibitor of EGFR (Ki/IC50: 5.2/29 pM, in cell-free assays) ; little inhibitory against FGFR, PGDFR, InsR, CSF-1 and Src.Smiles:
COC1=CC2=NC=NC(NC3=CC(Br)=CC=C3)=C2C=C1OCMolecular Formula:
C16H14BrN3O2Molecular Weight:
360.21Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
153436-54-5
