PD153035

CAT:
931-T2041-01
Size:
1 mL - 10 mM (in DMSO)
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
PD153035 - image 1

PD153035

  • Target:

    EGFR
  • Related Pathways:

    Angiogenesis|||JAK/STAT signaling|||Tyrosine Kinase/Adaptors
  • Purity:

    0.9931
  • Bioactivity:

    PD153035 (NSC-669364) hydrochloride is an effective and selective inhibitor of EGFR (Ki/IC50: 5.2/29 pM, in cell-free assays) ; little inhibitory against FGFR, PGDFR, InsR, CSF-1 and Src.
  • Smiles:

    COC1=CC2=NC=NC(NC3=CC(Br)=CC=C3)=C2C=C1OC
  • Molecular Formula:

    C16H14BrN3O2
  • Molecular Weight:

    360.21
  • Shipping Conditions:

    Cool pack
  • Storage Temperature:

    -20°C
  • CAS Number:

    153436-54-5