MRS 1523

• CAS Number :

  212329-37-8

• Target :

  Calcium Channel|||Adenosine Receptor|||Others

• Related Pathways :

  GPCR/G Protein|||Metabolism|||Neuroscience|||Others|||Membrane transporter/Ion channel

• Bioactivity :

  MRS 1523 can exert an antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons. MRS 1523 is an effective and selective adenosine A3 receptor antagonist Ki: 18.9 nM and 113 nM for human and rat A3 receptors, respectively) . In rat this corresponds to selectivities of 140- and 18-fold vs A1 and A2A receptors, respectively.

• Smiles :

  CCCOC(=O)c1c(CCC)c(C(=O)SCC)c(CC)nc1-c1ccccc1

• Molecular Formula :

  C23H29NO3S

• Molecular Weight :

  399.55

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C