FTI-2153

• Target:

  Others|||Transferase

• Related Pathways:

  Others|||Metabolism

• Bioactivity:

  FTI-2153 is a potent and highly selective farnesyltransferase (FTase) inhibitor (IC50: 1.4 nM) that is over 3000-fold more effective at blocking H-Ras (IC50: 10 nM) than Rap1A processing.

• Smiles:

  COC(=O)[C@H](CCSC)NC(=O)c1ccc(CNCc2cnc[nH]2)cc1-c1ccccc1C

• Molecular Formula:

  C25H30N4O3S

• Molecular Weight:

  466.6

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  344900-92-1