LS-75
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


LS-75
UNSPSC Description:
LS-75 is a PARP-1 inhibitor with blood-brain permeability and IC50 value of 18 μM. LS-75 has neuroprotective activity[1].Target Antigen:
PARPType:
Reference compoundRelated Pathways:
Cell Cycle/DNA Damage;EpigeneticsApplications:
Neuroscience-NeuromodulationField of Research:
Neurological DiseaseAssay Protocol:
https://www.medchemexpress.com/ls-75.htmlPurity:
99.31Smiles:
O=C1C2=CC=CC=C2NC=3N=CC=CC3N1Molecular Weight:
211.22References & Citations:
[1]André Schrattenholz, et al. Muscarinic antagonists with PARP and SIR modulating activity as agents for inflammatory diseases. US8039464B2.2011-10-18.Shipping Conditions:
Room TemperatureStorage Conditions:
4°C (Powder, protect from light)Clinical Information:
No Development ReportedCAS Number:
885-70-1
