GDC-0941 Dimethanesulfonate

• Catalog number
  9618-50
• Price
  Please ask
• Size
  50 mg

• Alternative_name
  4-[2-(1H-indazol-4-yl)-6-[(4-methylsulfonylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4-yl]morpholine;methanesulfonic acid; Pictilisib
• Description
  GDC-0941 is a potent, selective, inhibitor of pan-class I PI3 kinase (PI3K), with IC₅₀ values of 3, 33, 3, 75, 1230 and 580 nM for p110 α, β, δ and γ isoforms, DNA-PK and mTOR respectively. Displays antineoplastic activity.
• CAS Number
  957054-33-0
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₂₅H₃₅N₇O₉S₄
• Molecular Weight
  705.85
• Cell Permeable
  Yes
• Purity
  ≥98% by HPLC
• Solubilities
  DMSO (>10 mg/ml)
• Handling
  Protect from air and moisture
• Tag Line
  A potent, selective, inhibitor of pan-class I PI3 kinase
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• PubChem CID
  56972143
• PubChem CID Link
• SMILES
  CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6.CS(=O)(=O)O.CS(=O)(=O)O
• InChi
  InChI=1S/C23H27N7O3S2.2CH4O3S/c1-35(31,32)30-7-5-28(6-8-30)15-16-13-20-21(34-16)23(29-9-11-33-12-10-29)26-22(25-20)17-3-2-4-19-18(17)14-24-27-19;2*1-5(2,3)4/h2-4,13-14H,5-12,15H2,1H3,(H,24,27);2*1H3,(H,2,3,4)
• InChi Key
  RFRIKACSFOTIMU-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  GDC-0941   Dimethanesulfonate  
• Short name
  GDC-0941 Dimethanesulfonate
• Alternative name
  GDC-0941 Dimethanesulfonate

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