(R) -CE3F4

CAT: 0804-HY-108539A-01Size: 1 mgDry Ice: NoHazardous: No

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CAT#:0804-HY-108539A-01Size:1 mg

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Description

(R) -CE3F4 is a potent and selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1), with an IC50 of 4.2 μM, with 10-fold selectivity for Epac1 over Epac2 (IC50, 44 μM) . (R) -CE3F4 is more potent than racemic CE3F4 and (S) -CE3F4[1].

CAS Number

1593478-56-8

UNSPSC

12352005

Target

Ras

Type

Reference compound

Related Pathways

GPCR/G Protein; MAPK/ERK Pathway

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/r-ce3f4.html

Purity

99.3

Solubility

DMSO : ≥ 50 mg/mL

Smiles

O=CN1[C@H](C)CCC2=C1C=C(Br)C(F)=C2Br

Molecular Formula

C11H10Br2FNO

Molecular Weight

351.01

References & Citations

[1]Courilleau D, et al. The (R) -enantiomer of CE3F4 is a preferential inhibitor of human exchange protein directly activated by cyclic AMP isoform 1 (Epac1) . Biochem Biophys Res Commun. 2013 Oct 25;440 (3) :443-8.

Shipping Conditions

Blue Ice

Storage Conditions

-20°C, 3 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

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B4927-25	CE3F4
T12616-01	(R) -CE3F4
A20067-10	CE3F4 10mg
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A20067-100	CE3F4 100mg
A20067-25	CE3F4 25mg
A20067-50	CE3F4 50mg
A20067-5	CE3F4 5mg

(R) -CE3F4

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