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Tegoprazan (Benzoate)

CAT: 0804-HY-17623DSize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-17623DSize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Tegoprazan Benzoate is the benzoate form of Tegoprazan. Tegoprazan (CJ-12420), a potassium-competitive acid blocker, is a potent, oral active and highly selective inhibitor of gastric H+/K+-ATPase that could control gastric acid secretion and motility, with IC50 values ranging from 0.29-0.52 μM for porcine, canine, and human H+/K+-ATPases in vitro[1].
Product Name Alternative
CJ-12420 (Benzoate) ; RQ-00000004 (Benzoate)
UNSPSC
12352005
Target
Proton Pump
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/tegoprazan-benzoate.html
Solubility
10 mM in DMSO
Smiles
FC1=CC(F)=C2[C@@H](OC3=CC(C(N(C)C)=O)=CC4=C3N=C(C)N4)CCOC2=C1.O=C(O)C5=CC=CC=C5
Molecular Formula
C27H25F2N3O5
Molecular Weight
509.50
References & Citations
[1]Takahashi N, et al. Tegoprazan, a Novel Potassium-Competitive Acid Blocker to Control Gastric Acid Secretion and Motility. J Pharmacol Exp Ther. 2018 Feb;364 (2) :275-286.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 4

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