GPS1573

CAT: 0804-HY-P10571-01Size: 1 mgDry Ice: NoHazardous: No

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CAT#:0804-HY-P10571-01Size:1 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Description

GPS1573 is a noncompetitive antagonist of melanocortin type 2 receptor (MC2R) that dose-dependently antagonizes ACTH-stimulated MC2R activity (IC50=66 nM) . GPS1573 can be used in the study of Cushing's disease due to its highly selective antagonism of MC2R[1].

CAS Number

2445822-54-6

UNSPSC

12352209

Target

Melanocortin Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Endocrinology

Assay Protocol

https://www.medchemexpress.com/gps1573.html

Purity

99.31

Smiles

O=C(N1[C@@H](CCC1)C(N[C@H](CC2=CC=CC=C2)C(N[C@@H](CCCNC(N)=N)C(N[C@H](CC3=CNC4=CC=CC=C34)C(N[C@@H](CC5=CC=CC=C5)C(N[C@@H](CCCCN)C(N[C@@H](C)C(N[C@@H](C(C)C)C(NCC(N[C@@H](CCCCN)C(N[C@@H](CCCCN)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CCCNC(N)=N)C(N)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)[C@H](CCCC)N

Molecular Formula

C86H138N28O14

Molecular Weight

1788.20

References & Citations

[1]Bouw E, et al. Development of potent selective competitive-antagonists of the melanocortin type 2 receptor[J]. Molecular and Cellular Endocrinology, 2014, 394 (1-2) : 99-104.

Shipping Conditions

Blue Ice

Storage Conditions

-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)

Scientific Category

Peptides

Clinical Information

No Development Reported

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GPS1573

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