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GSK2807

CAT: 0804-HY-104009Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-104009Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GSK2807 is a potent and selective SAM-competitive inhibitor of SMYD3, exhibiting a Ki value of 14 nM, and it may be useful for cancer treatment by preventing the methylation of MEKK2.
CAS Number
2245255-65-4
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gsk2807.html
Smiles
NC1=C(N=CN2[C@@H]3O[C@H](CN(CC[C@H](N)C(O)=O)CCCN(C)C)[C@@H](O)[C@H]3O)C2=NC=N1
Molecular Formula
C19H32N8O5
Molecular Weight
452.51
References & Citations
[1]Structure-Based Design of a Novel SMYD3 Inhibitor that Bridges the SAM-and MEKK2-Binding Pockets
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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