Products for Research Use Only
RegisterLogin

GSK217

CAT: 0804-HY-153242Size: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-153242Size:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
GSK217 is a potent, selective, and highly soluble bromo and extraterminal domain (BET) second bromodomain (BD2) inhibitor. GSK217 can be used for the research of oncology and immune inflammation research[1].
CAS Number
2748687-92-3
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/gsk217.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC(C2=CN(C)N=N2)=NC(CC3=C4C=CNC4=CC=C3)=C1)NCC
Molecular Formula
C20H20N6O
Molecular Weight
360.41
References & Citations
[1]Aylott HE, et al. Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors. J Med Chem. 2021 Mar 25;64 (6) :3249-3281.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-136555-01GSK717
HY-132296-01GSK215
HY-18948-01GSK321
HY-132880-01GSK251
HY-118316GSK223
HY-148631GSK137
HY-132232GSK097
HY-176709GSK147
HY-104009GSK2807
HY-114492-01GSK547

Alternative Products

CatalogName
T79018-01GSK217

Popular Products