hCYP3A4 Fluorogenic substrate 1

CAT:

804-HY-155002-06

Size:

10 mM / 1 mL

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CAS Number: 186299-00-3
UNSPSC Description: hCYP3A4 Fluorogenic substrate 1 is a potrnt hCYP3A4 fluorogenic substrate with an Km value of 0.36 μM. hCYP3A4 Fluorogenic substrate 1 can be used for cell and in vivo imaging[1].
Target Antigen: Cytochrome P450
Type: Reference compound
Related Pathways: Metabolic Enzyme/Protease
Applications: Metabolism-sugar/lipid metabolism
Field of Research: Metabolic Disease
Assay Protocol: https://www.medchemexpress.com/hcyp3a4-fluorogenic-substrate-1.html
Solubility: DMSO : 12.5 mg/mL (ultrasonic;warming;heat to 60°C)
Smiles: O=C(C1=C2C(C3=O)=CC=CC2=CC=C1)N3CC4=CC=C(F)C=C4
Molecular Weight: 305.30
References & Citations: [1]He RJ, et al. Rationally Engineered CYP3A4 Fluorogenic Substrates for Functional Imaging Analysis and Drug-Drug Interaction Studies. J Med Chem. 2023 May 25;66(10):6743-6755.
Shipping Conditions: Room Temperature
Clinical Information: No Development Reported

Cat	Name
HY-155002-06	hCYP3A4 Fluorogenic substrate 1
HY-155002-05	hCYP3A4 Fluorogenic substrate 1
HY-155002-04	hCYP3A4 Fluorogenic substrate 1
HY-155002-03	hCYP3A4 Fluorogenic substrate 1
HY-155002-02	hCYP3A4 Fluorogenic substrate 1
HY-155002-01	hCYP3A4 Fluorogenic substrate 1
HY-D2284-01	SGPL1 fluorogenic substrate
HY-D2284-02	SGPL1 fluorogenic substrate
HY-P10189	α-Secretase Substrate, Fluorogenic
HY-P10073	Calpain-1 substrate, fluorogenic

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