Products for Research Use Only

SMARCA2-IN-9

CAT: 0804-HY-161881Size: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-161881Size:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
SMARCA2-IN-9 (compound 11) is a SMARCA2, PBRM1 bromodomains 2 (PBRM1 (2) ), and PBRM1 bromodomains 5 (PBRM1 (5) ) inhibitor with Kd values of 1.6 μM, 2.5 μM, and 3.95 μM, respectively[1].
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/smarca2-in-9.html
Smiles
NC1=C(C2=CC=CC=C2)C=C(C3=CC=CO3)N=N1
Molecular Formula
C14H11N3O
Molecular Weight
237.26
References & Citations
[1]Andrea G Cochran, et al. GNE-235: A Lead Compound Selective for the Second Bromodomain of PBRM1. J Med Chem. 2023 Sep 28;66 (18) :13116-13134.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported