Apalutamide-d4

CAT: 0804-HY-16060S-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0804-HY-16060S-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Apalutamide-d4 is a deuterium labeled Apalutamide. Apalutamide is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM[1].
CAS Number
[1638885-65-0]
Product Name Alternative
ARN-509-d4
UNSPSC
12352005
Target
Androgen Receptor
Type
Isotope-Labeled Compounds
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Purity
99.90
Solubility
DMSO : 50mg/mL (ultrasonic) |H2O
Smiles
O=C(NC)C1=CC=C(N(C(N(C2=CC(C(F)(F)F)=C(C#N)N=C2)C3=O)=S)C43C([2H])([2H])CC4([2H])[2H])C=C1F
Molecular Formula
C21H11D4F4N5O2S
Molecular Weight
481.46
References & Citations
[1]Clegg NJ, et al. ARN-509: a novel antiandrogen for prostate cancer treatment. Cancer Res. 2012 Mar 15;72 (6) :1494-503.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported

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