DA 4626

• Description :

  DA 4626 is a competitive H2-histamine receptor antagonist. DA 4626 inhibits adenylate cyclase activity with a KB value of 40 nM[1].

• UNSPSC :

  12352005

• Target :

  Adenylate Cyclase; Histamine Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

• Applications :

  Metabolism-protein/nucleotide metabolism

• Field of Research :

  Metabolic Disease

• Assay Protocol :

  https://www.medchemexpress.com/da-4626.html

• Smiles :

  CC(/N=C/NC1=CC=C(C2=CN=CN2)C=C1)(C)C

• Molecular Formula :

  C14H18N4

• Molecular Weight :

  242.32

• References & Citations :

  [1]Micheletti R, et al. Evaluation of novel compounds interacting with H2-histamine receptors: effect on histamine-sensitive adenylate cyclase activity in guinea-pig gastric mucosa. Agents Actions. 1985 Jul;16 (5) :291-4.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• Isoform :

  H2 Receptor

• CAS Number :

  [83184-14-9]