KDM4-IN-3
CAT:
804-HY-132896-02
Size:
100 mg
Price:
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
KDM4-IN-3
- CAS Number: 1068515-53-6
- UNSPSC Description: KDM4-IN-3 is a KDM4 inhibitor that exhibits improved potency in biochemical assays, is cell-permeable, and kills prostate cancer cells at low micromolar concentrations.
- Target Antigen: Histone Demethylase
- Type: Reference compound
- Related Pathways: Epigenetics
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/kdm4-in-3.html
- Purity: 99.36
- Solubility: DMSO : 116.67 mg/mL (ultrasonic)
- Smiles: OC1=C(C2=CC=CC=C2)C(C)=NN1C3=NC4=CC=CC=C4N3
- Molecular Weight: 290.32
- References & Citations: [1]Carter DM, et al. Enhanced Properties of a Benzimidazole Benzylpyrazole Lysine Demethylase Inhibitor: Mechanism-of-Action, Binding Site Analysis, and Activity in Cellular Models of Prostate Cancer. J Med Chem. 2021 Oct 14;64(19):14266-14282.
- Shipping Conditions: Room Temperature
- Storage Conditions: -20°C, 3 years; 4°C, 2 years (Powder)
- Clinical Information: No Development Reported