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Taltirelin-13C, d3

CAT: 0804-HY-B0596SSize: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-B0596SSize:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Taltirelin-13C, d3 (TA-0910-13C, d3) is 13C and deuterated labeled Taltirelin. Taltirelin (TA0910) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Product Name Alternative
TA-0910-13C, d3
UNSPSC
12352005
Target
Apoptosis; Isotope-Labeled Compounds; Thyroid Hormone Receptor
Type
Isotope-Labeled Compounds
Related Pathways
Apoptosis; Others; Vitamin D Related/Nuclear Receptor
Applications
Neuroscience-Neuromodulation
Field of Research
Endocrinology; Neurological Disease
Solubility
10 mM in DMSO
Smiles
O=C(N(CCC1)[C@@H]1C(N)=O)[C@@H](NC([C@@H](NC2=O)CC(N2[13C]([2H])([2H])[2H])=O)=O)CC3=CN=CN3
Molecular Formula
C16 13CH20D3N7O5
Molecular Weight
409.42
References & Citations
[1]Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne) . 2012 Oct 9;3:120.|[2]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53 (2) :211-216.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported

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