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DDR1-IN-8

CAT: 0804-HY-162102Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-162102Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
DDR1-IN-8 (compound 7s) is a potent inhibitor of DDR1/2, with the IC50 values of 0.045 μM and 0.126 μM, respectively. DDR1-IN-8 has anti-tumor activity[1].
CAS Number
3038810-92-0
UNSPSC
12352005
Target
Discoidin Domain Receptor
Type
Reference compound
Related Pathways
Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ddr1-in-8.html
Solubility
10 mM in DMSO
Smiles
O=C(NCC1=CN(CC(N2CCN(CC2)C)=O)C3=C1C=C(F)C=C3)NC4=CC=C(C=C4F)F
Molecular Formula
C23H24F3N5O2
Molecular Weight
459.46
References & Citations
[1]Shangke Liu, et al. Design, synthesis, and biological evaluation of novel discoidin domain receptor inhibitors for the treatment of lung adenocarcinoma and pulmonary fibrosis. Eur J Med Chem. 2024 Feb 5:265:116100.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
DDR1; DDR2

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