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DYRK2-IN-1

CAT: 0804-HY-161014Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-161014Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
DYRK2-IN-1 (Compd 54) is an orally bioavailable DYRK2 inhibitor, with an IC50 of 14 nM. DYRK2-IN-1 (Compd 54) can be used in the study of prostate cancer[1].
UNSPSC
12352005
Target
DYRK
Type
Reference compound
Related Pathways
Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/dyrk2-in-1.html
Solubility
10 mM in DMSO
Smiles
FC1=CN=C(N=C1C2=CC=C3N=C(SC3=C2)N(CC)CC)NC4=NC=C(C=C4)C(N5CCN(CC5)C(C6CC6)=O)=O
Molecular Formula
C29H31FN8O2S
Molecular Weight
574.67
References & Citations
[1]Kai Yuan, et al. Discovery of Potent, Selective, and Orally Bioavailable DYRK2 Inhibitors for the Treatment of Prostate Cancer. J Med Chem. 2023 Dec 14;66 (23) :16235-16256.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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