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DYRKs-IN-2

CAT: 0804-HY-128759Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-128759Size:1 Each
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Description
DYRKs-IN-2 (Example 132) is a potent DYRKs inhibitor with IC50s of 30.6 nM and 12.8 nM for DYRK1B and DYRK1A, respectively. DYRKs-IN-2 has antitumor activity[1].
CAS Number
1386980-04-6
UNSPSC
12352005
Target
DYRK
Type
Reference compound
Related Pathways
Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/dyrks-in-2.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC2=CN=C(NCCCN3CCN(C)CC3)N=C2NC1=O)NC4=CC(C(NC(C5=CC=CC=C5)CCN)=O)=CC=C4Cl
Molecular Formula
C32H38ClN9O3
Molecular Weight
632.16
References & Citations
[1]Kevin Anderson, et al. Pyrido pyrimidines. US20120184542A1
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
DYRK1

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