KCC2 Modulator-1

• Description:

  KCC2 Modulator-1 (Example 52) is a KCC2 modulator with an EC50 value of 0.146 μM. KCC2 Modulator-1 can be used for the research of KCC2 mediated diseases[1].

• UNSPSC:

  12352005

• Target:

  Potassium Channel

• Type:

  Reference compound

• Related Pathways:

  Membrane Transporter/Ion Channel

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer; Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/kcc2-modulator-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C1C2=C(CN1C(C)C)C(NC3=CC=C(C4=CC=C(OCCCCCC#C)C=C4)C=C3)=NC(N5CCOC(C6CC6)C5)=N2

• Molecular Formula:

  C35H41N5O3

• Molecular Weight:

  579.73

• References & Citations:

  [1]Rebecca Elizabeth Jarvis, et al. Fused pyrimidine compounds as kcc2. Patent. WO2021180952 A1.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  [2704531-36-0]