SORT-PGRN interaction inhibitor 3
CAT:
804-HY-153688
Size:
Inquire
Price:
Ask
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

SORT-PGRN interaction inhibitor 3
- CAS Number: 2691846-87-2
- UNSPSC Description: SORT-PGRN interaction inhibitor 3 (Compound 13) is a SORT-PGRN interaction inhibitor (IC50: 0.17 μM). SORT-PGRN interaction inhibitor 3 can be used for research of neurodegenerative diseases[1].
- Target Antigen: Neurotensin Receptor
- Type: Reference compound
- Related Pathways: GPCR/G Protein;Neuronal Signaling
- Applications: Neuroscience-Neurodegeneration
- Field of Research: Neurological Disease
- Assay Protocol: https://www.medchemexpress.com/sort-pgrn-interaction-inhibitor-3.html
- Solubility: 10 mM in DMSO
- Smiles: CC(C)(C)CC[C@@H](C(O)=O)NC(C1=CC(Cl)=CC(Cl)=C1)=O
- Molecular Weight: 332.22
- References & Citations: [1]Stachel SJ, et al. Identification of potent inhibitors of the sortilin-progranulin interaction. Bioorg Med Chem Lett. 2020 Sep 1;30(17):127403.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported