FAAH/cPLA2α-IN-1

FAAH/cPLA2α-IN-1

• CAS Number: 1696401-38-3
• UNSPSC Description: FAAH/cPLA2α-IN-1 is a dual inhibitor of FAAH and cPLA2α with IC50s of 32 and 47 nM, respectively[1].
• Target Antigen: FAAH; Phospholipase
• Type: Reference compound
• Related Pathways: Metabolic Enzyme/Protease;Neuronal Signaling
• Applications: COVID-19-immunoregulation
• Field of Research: Inflammation/Immunology; Neurological Disease
• Assay Protocol: https://www.medchemexpress.com/faah-cpla2α-in-1.html
• Solubility: 10 mM in DMSO
• Smiles: O=C(CCC1=NN(CC(COC2=CC=C(C=C2)OCCCCCC)=O)N=N1)O
• Molecular Weight: 390.43
• References & Citations: [1]Ekodo Voundi M, et al. Synthesis, activity and metabolic stability of propan-2-one substituted tetrazolylalkanoic acids as dual inhibitors of cytosolic phospholipase A2α and fatty acid amide hydrolase. RSC Med Chem. 2023 Aug 10;14(10):2079-2088.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported