Adenosine receptor inhibitor 2

CAT:

804-HY-147908

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CAS Number: 2550401-76-6
UNSPSC Description: Adenosine receptor inhibitor 2 (compound 14b) is a potent AR (adenosine receptor) inhibitor. Adenosine receptor inhibitor 2 shows dual affinity toward A1/A2A ARs with higher affinity for the A1- than the A2AAR. Adenosine receptor inhibitor 2 has Ki values of 52.2 nM for the A1AR and 167 nM for the A2AAR[1].
Target Antigen: Adenosine Receptor
Type: Reference compound
Related Pathways: GPCR/G Protein
Applications: COVID-19-immunoregulation
Field of Research: Inflammation/Immunology
Assay Protocol: https://www.medchemexpress.com/adenosine-receptor-inhibitor-2.html
Solubility: 10 mM in DMSO
Smiles: O=C(N1CC)N(CC)C2=C(N(C)C(NCC3=CC=CC(Br)=C3)=N2)C1=O
Molecular Weight: 406.28
References & Citations: [1]Załuski M, et al. 8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation. Bioorg Chem. 2020 Aug;101:104033.
Shipping Conditions: Room temperature
Clinical Information: No Development Reported

Cat	Name
HY-147908	Adenosine receptor inhibitor 2
HY-147907-03	Adenosine receptor inhibitor 1
HY-147907-01	Adenosine receptor inhibitor 1
HY-147907-02	Adenosine receptor inhibitor 1
HY-162851	Adenosine receptor agonist 1
HY-W063197-03	Adenosine receptor antagonist 4
HY-144419-05	Adenosine receptor antagonist 3
HY-141865	Adenosine receptor antagonist 1
HY-162787	Adenosine receptor antagonist 5
HY-W063197-02	Adenosine receptor antagonist 4

Cat	Name
T61850-50mg	Adenosine receptor inhibitor 1
T62018-1g	Adenosine receptor inhibitor 2
T62018-50mg	Adenosine receptor inhibitor 2
T61850-10mg	Adenosine receptor inhibitor 1
T61850-5mg	Adenosine receptor inhibitor 1
T62018-5mg	Adenosine receptor inhibitor 2
T62018-10mg	Adenosine receptor inhibitor 2
T61850-1g	Adenosine receptor inhibitor 1
T61850-1mg	Adenosine receptor inhibitor 1
T62018-1mg	Adenosine receptor inhibitor 2