Adenosine receptor inhibitor 1
CAT:
804-HY-147907-03
Size:
10 mg
Price:
Ask
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
Adenosine receptor inhibitor 1
- CAS Number: 2550400-52-5
- UNSPSC Description: Adenosine receptor inhibitor 1 is a potent and selective adenosine receptor (AR) inhibitor with Ki values of >1000, 68.5, >1000, >1000 nM for A1AR, A2AAR, A2BAR, A3AR, respectively. Adenosine receptor inhibitor 1 shows antinociceptive activity, anti-inflammatory effect and peripheral analgesic effect. Adenosine receptor inhibitor 1 has the potential for the research of cancer or neurodegenerative diseases[1].
- Target Antigen: Adenosine Receptor
- Type: Reference compound
- Related Pathways: GPCR/G Protein
- Field of Research: Cancer; Inflammation/Immunology; Neurological Disease
- Assay Protocol: https://www.medchemexpress.com/adenosine-receptor-inhibitor-1.html
- Solubility: 10 mM in DMSO
- Smiles: O=C(N1CC)N(C)C2=C(N(C)C(NCC3=C(Cl)C=CC(OC)=C3F)=N2)C1=O
- Molecular Weight: 395.82
- References & Citations: [1]Załuski M, et al. 8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation. Bioorg Chem. 2020 Aug;101:104033.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported