Adenosine receptor antagonist 1

• UNSPSC Description:

  Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aR than A2bR.

• Target Antigen:

  Adenosine Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/adenosine-receptor-antagonist-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  NC1=NC(C2=CC=CC=C2)=C(C3=NC(CC4=C(C=C(C=N4)F)Cl)=NN13)C5=CNC(C=C5)=O

• Molecular Weight:

  447.85

• References & Citations:

  [1]Lamb ML, et al. Triazole compounds as adenosine receptor antagonists. WO2021156439A1.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  2682930-40-9