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MGAT3/4-IN-2

CAT: 0804-HY-146281Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-146281Size:1 Each
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Description
MGAT3/4-IN-2 (compound 27b) is a potent mGAT3/mGAT4 inhibitor, with pIC50 values of 5.44 and 5.25, respectively[1].
CAS Number
2556833-68-0
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/mgat3-4-in-2.html
Solubility
10 mM in DMSO
Smiles
CC1=C(SC=C1)/C(C2=C(C=CS2)C)=C\CCN(C(C(NCC3=C(C=CC=C3)Cl)=O)CCN)C
Molecular Formula
C26H32ClN3OS2
Molecular Weight
502.13
References & Citations
[1]Zaręba P, et al. Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice. Eur J Med Chem. 2020 Feb 15;188:111920.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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