Elastase-IN-1

• Description :

  Elastase-IN-1 (Compound Q11) is an elastase inhibitor with an IC50 of 0.897 µM. Elastase-IN-1 is non-toxic[1].

• UNSPSC :

  12352005

• Target :

  Elastase

• Type :

  Reference compound

• Related Pathways :

  Metabolic Enzyme/Protease

• Applications :

  COVID-19-immunoregulation

• Field of Research :

  Cancer; Inflammation/Immunology

• Assay Protocol :

  https://www.medchemexpress.com/elastase-in-1.html

• Solubility :

  10 mM in DMSO

• Smiles :

  O=C(N/N=C/C1=NC2=CC=CC=C2C=C1)C3=CC=C([N+]([O-])=O)C=C3

• Molecular Formula :

  C17H12N4O3

• Molecular Weight :

  320.30

• References & Citations :

  [1]Vanjare BD, et al. Elastase inhibitory activity of quinoline Analogues: Synthesis, kinetic mechanism, cytotoxicity, chemoinformatics and molecular docking studies. Bioorg Med Chem. 2022 Jun 1;63:116745.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• CAS Number :

  [678152-73-3]