Elastase-IN-1
CAT:
804-HY-146070
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

Elastase-IN-1
- CAS Number: 678152-73-3
- UNSPSC Description: Elastase-IN-1 (Compound Q11) is an elastase inhibitor with an IC50 of 0.897 µM. Elastase-IN-1 is non-toxic[1].
- Target Antigen: Elastase
- Type: Reference compound
- Related Pathways: Metabolic Enzyme/Protease
- Applications: COVID-19-immunoregulation
- Field of Research: Cancer; Inflammation/Immunology
- Assay Protocol: https://www.medchemexpress.com/elastase-in-1.html
- Solubility: 10 mM in DMSO
- Smiles: O=C(N/N=C/C1=NC2=CC=CC=C2C=C1)C3=CC=C([N+]([O-])=O)C=C3
- Molecular Weight: 320.30
- References & Citations: [1]Vanjare BD, et al. Elastase inhibitory activity of quinoline Analogues: Synthesis, kinetic mechanism, cytotoxicity, chemoinformatics and molecular docking studies. Bioorg Med Chem. 2022 Jun 1;63:116745.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported