Products for Research Use Only
RegisterLogin

CPI-4203

CAT: 0804-HY-123419Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-123419Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
CPI-4203 is a potent KDM5A inhibitor with an IC50 of 250 nM. CPI-4203 is competitive with 2-oxoglutarate (2-OG). CPI-4203 is structurally related to CPI-455 but is less potent[1].
CAS Number
1628214-07-2
UNSPSC
12352005
Target
Histone Demethylase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/cpi-4203.html
Purity
99.0
Solubility
DMSO : 25 mg/mL (ultrasonic; warming)
Smiles
N#CC1=C(N2N=C1)NC(C3=C(C=CC=C3)C)=C(C2=O)CC
Molecular Formula
C16H14N4O
Molecular Weight
278.31
References & Citations
[1]Vinogradova M, et al. An inhibitor of KDM5 demethylases reduces survival of drug-tolerant cancer cells. Nat Chem Biol. 2016 Jul;12 (7) :531-8.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-145654MRS-4203
HY-15955CPI-360
HY-15956ACPI-169
HY-15846-01CPI-203
HY-100482-01CPI-637
HY-100421-01CPI-455
HY-136285-01CPI-1612
HY-111085CPI-905
HY-134899CPI-1328
HY-100376-01CPI-1189

Alternative Products

CatalogName
BA4802-5CPI-4203
DQC21407-01CPI 4203
A16177-100CPI 4203 100mg
A16177-5CPI 4203 5mg
A16177-10CPI 4203 10mg
A16177-25CPI 4203 25mg
A16177-50CPI 4203 50mg
BU167832-01UNC 4203
MBS5680488-01Anti-h NGAL 4203 SPTN-5
B1081-5CPI-203

Popular Products