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A-123189

CAT: 0804-HY-116623Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-116623Size:1 Each
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Description
A-123189 is a selective and potent α1D antagonist with Kis of 0.312 and 0.17 for human α1D and rat α1D, respectively. A-123189 displays selectivities between 10- to 20-fold for the α1D receptor over the human α1A and rat α1A receptors[1].
CAS Number
255713-53-2
UNSPSC
12352005
Target
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/a-123189.html
Solubility
10 mM in DMSO
Smiles
O=C1N(C(C2=C(N1)SC=C2C3=CC=CC(C)=C3)=O)CCN4CCN(CC4)C5=CC=CC=C5OC
Molecular Formula
C26H28N4O3S
Molecular Weight
476.59
References & Citations
[1]K P Briski, et al. Antagonism of type II, but not type I glucocorticoid receptors results in elevated basal luteinizing hormone release in male rats. Bioorganic & Medicinal Chemistry Letters, Volume 11, Issue 9, 7 May 2001, Pages 1119-1121.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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