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SSTR5 antagonist 2 (TFA)

CAT: 0804-HY-114191ASize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-114191ASize:1 Each
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Description
SSTR5 Antagonist 1 (compound 10) is a highly potent, oral active and selective somatostatin (receptor) subtype 5 (SSTR5) antagonist and has potential for the research of treat type 2 diabetes mellitus (T2DM) [1].
CAS Number
1254733-98-6
UNSPSC
12352005
Target
Somatostatin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease; Endocrinology
Assay Protocol
https://www.medchemexpress.com/sstr5-antagonist-2-tfa.html
Solubility
10 mM in DMSO
Smiles
FC(C=C1)=CC=C1C2=C(OCC)C=C(CN3CCC4(CN(C5=CC=C(C(O)=O)C=C5)C(C4)=O)CC3)C=C2OCC.OC(C(F)(F)F)=O
Molecular Formula
C34H36F4N2O7
Molecular Weight
660.65
References & Citations
[1]Liu W, et al. Discovery and Pharmacology of a Novel Somatostatin Subtype 5 (SSTR5) Antagonist: Synergy with DPP-4 Inhibition. ACS Med Chem Lett. 2018 Sep 12;9 (11) :1082-1087.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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