GV-150013

• UNSPSC Description:

  GV-150013 is a selective CCK-B receptor antagonist. GV-150013 has sleep aid effect[1].

• Target Antigen:

  Cholecystokinin Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;Neuronal Signaling

• Field of Research:

  Others

• Assay Protocol:

  https://www.medchemexpress.com/gv-150013.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C([C@@H](C1=O)NC(NC2=CC=CC=C2)=O)N(C3=CC=CC=C3)C4=CC=CC=C4N1CC56CC7CC(CC(C7)C6)C5

• Molecular Weight:

  534.65

• References & Citations:

  [1]Crespi F. Cholecystokinin-B (CCK-B) receptor antagonists improve "aged" sleep: a new class of sleep modulators? Methods Find Exp Clin Pharmacol. 1999 Jan-Feb;21(1):31-8.|[2]F.Crespi, et al. Influence of cholecystokinin-B (CCK-B) receptor antagonists on rat electroencephalography (EEG): A new class of sleep modulators? Gaviraghi. Dept of Pharmacology GlaxoWellcome S.p.A., Medicine Research Centre, via A. Fleming, 4, 37135 Verona, Italy

• Shipping Conditions:

  Room temperature

• Clinical Information:

  Phase 2

• CAS Number:

  167355-22-8