GV-150013

• Description :

  GV-150013 is a selective CCK-B receptor antagonist. GV-150013 has sleep aid effect[1].

• UNSPSC :

  12352005

• Target :

  Cholecystokinin Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Neuronal Signaling

• Field of Research :

  Others

• Assay Protocol :

  https://www.medchemexpress.com/gv-150013.html

• Solubility :

  10 mM in DMSO

• Smiles :

  O=C([C@@H](C1=O)NC(NC2=CC=CC=C2)=O)N(C3=CC=CC=C3)C4=CC=CC=C4N1CC56CC7CC(CC(C7)C6)C5

• Molecular Formula :

  C33H34N4O3

• Molecular Weight :

  534.65

• References & Citations :

  [1]Crespi F. Cholecystokinin-B (CCK-B) receptor antagonists improve "aged" sleep: a new class of sleep modulators? Methods Find Exp Clin Pharmacol. 1999 Jan-Feb;21 (1) :31-8.|[2]F.Crespi, et al. Influence of cholecystokinin-B (CCK-B) receptor antagonists on rat electroencephalography (EEG) : A new class of sleep modulators? Gaviraghi. Dept of Pharmacology GlaxoWellcome S.p.A., Medicine Research Centre, via A. Fleming, 4, 37135 Verona, Italy

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  Phase 2

• CAS Number :

  [167355-22-8]