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Tabimorelin (hemifumarate)

CAT: 0804-HY-103540-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-103540-01Size:1 mg
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Description
Tabimorelin (NN703) hemifumarate is an orally active growth hormone (GH) secretagogue. Tabimorelin hemifumarate is also a potent inhibitor of CYP3A4 activity[1].
CAS Number
242143-80-2
Product Name Alternative
NN703 (hemifumarate)
UNSPSC
12352005
Target
Cytochrome P450
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/tabimorelin-hemifumarate.html
Solubility
10 mM in DMSO
Smiles
CNC([C@@H](CC1=CC=CC=C1)N(C)C([C@H](N(C)C(/C=C/CC(C)(N)C)=O)CC2=CC3=CC=CC=C3C=C2)=O)=O.OC(/C=C/C(O)=O)=O
Molecular Formula
C32H40N4O3.1/2C4H4O4
Molecular Weight
586.72
References & Citations
[1]Zdravkovic M, et al. A clinical study investigating the pharmacokinetic interaction between NN703 (tabimorelin), a potential inhibitor of CYP3A4 activity, and midazolam, a CYP3A4 substrate. Eur J Clin Pharmacol. 2003 Feb;58 (10) :683-8.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CYP3