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GR125487 (sulfamate)

CAT: 0804-HY-103146Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-103146Size:1 Each
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Description
GR125487 sulfamate is an orally active and selective antagonist of 5-HT4R. GR125487 sulfamate effectively blocks the cognition enhancing effect. GR125487 sulfamate can be used to study memory disorders, gastrointestinal disorders, mood disorders and urinary tract dysfunction[1].
CAS Number
859502-43-5
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/gr125487-sulfamate.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=C(NC2=C1C=C(F)C=C2)OC)OCC3CCN(CC3)CCNS(=O)(C)=O.O=S(O)(N)=O
Molecular Formula
C19H29FN4O8S2
Molecular Weight
524.58
References & Citations
[1]Nirogi, R., et al. Synthesis of GR 125487, a selective 5-HT4receptor antagonist. Synthetic Communications, 46 (12), 1036–1043.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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