Azaperone-d4

• Description:

  Azaperone-d4 is the deuterium labeled Azaperone. Azaperone (R-1929) acts as a dopamine antagonist but also has some antihistaminic and anticholinergic properties. Azaperone is a pyridinylpiperazine and butyrophenone neuroleptic agent with antiemetic effects, which is used mainly as a tranquilizer in veterinary medicine.

• Product Name Alternative:

  R-1929-d4

• UNSPSC:

  12352005

• Hazard Statement:

  H301

• Target:

  Dopamine Receptor; Isotope-Labeled Compounds

• Type:

  Isotope-Labeled Compounds

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling; Others

• Field of Research:

  Neurological Disease

• Purity:

  98.16

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(C1=C([2H])C([2H])=C(C([2H])=C1[2H])F)CCCN2CCN(C3=CC=CC=N3)CC2

• Molecular Formula:

  C19H18D4FN3O

• Molecular Weight:

  331.42

• Precautions:

  H301

• References & Citations:

  [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216.

• Shipping Conditions:

  Blue Ice

• Storage Conditions:

  -20°C, 3 years (Powder)

• Scientific Category:

  Isotope-Labeled Compounds

• Clinical Information:

  No Development Reported

• CAS Number:

  [1173021-72-1]