SER-601

• Description:

  SER-601 is a potent and selective peripheral cannabinoid (CB2) receptor agonist with a Ki of 6.3 nM. SER-601 has analgesic and antidiabetic properties and can be used for relevant research[1].

• UNSPSC:

  12352005

• Target:

  Cannabinoid Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/ser-601.html

• Smiles:

  O=C(C(C(C1=CC(C(C)C)=CC=C12)=O)=CN2CCCCC)NC3(C[C@@H](C4)C5)C[C@@H]5C[C@@H]4C3

• Molecular Formula:

  C28H38N2O2

• Molecular Weight:

  434.61

• References & Citations:

  [1]Pasquini S, et al. Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J Med Chem. 2008 Aug 28;51 (16) :5075-84.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  1048038-90-9