AURKA-IN-1
CAT:
804-HY-161407
Size:
Inquire
Price:
Ask
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

AURKA-IN-1
- UNSPSC Description: AURKA-IN-1 (compound 9) is an cell-active covalent AURKA inhibitor. AURKA-IN-1 is a lysine-reactive activity probe[1].
- Target Antigen: Aurora Kinase
- Type: Reference compound
- Related Pathways: Cell Cycle/DNA Damage;Epigenetics
- Applications: Cancer-Kinase/protease
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/aurka-in-1.html
- Solubility: 10 mM in DMSO
- Smiles: O=C(NCC#C)C1=CC(NC2=NNC(C3CC3)=C2)=NC(N4CCN(C(C5=CC=C(OS(=O)(F)=O)C=C5)=O)CC4)=N1
- Molecular Weight: 568.58
- References & Citations: [1]Guanghui Tang, et al. Global Reactivity Profiling of the Catalytic Lysine in Human Kinome for Covalent Inhibitor Development. Angew Chem Int Ed Engl. 2024, 63, 12.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported