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Carvedilol Glucuronide

CAT: 0804-HY-137387-01Size: 500 µgDry Ice: NoHazardous: No
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CAT#:0804-HY-137387-01Size:500 µg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Carvedilol Glucuronide is the metabolite of Carvedilol. Carvedilol (BM 14190) is an antagonist for β/α-1 adrenergic receptor. Carvedilol inhibits lipid peroxidation with an IC50 of 5 μM. Carvedilol is an antihypertensive agent with potential use in angina and congestive heart failure. Carvedilol is an autophagy inducer that inhibits the NLRP3 inflammasome[1].
CAS Number
114869-83-9
UNSPSC
12352005
Target
Drug Metabolite
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Others; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/carvedilol-glucuronide.html
Smiles
OC([C@@H](O[C@H]1OC(COC2=C3C4=CC=CC=C4NC3=CC=C2)CNCCOC5=C(OC)C=CC=C5)[C@@H](O)[C@H](O)[C@H]1O)=O
Molecular Formula
C30H34N2O10
Molecular Weight
582.60
References & Citations
[1]Hanioka N, et al., Stereoselective glucuronidation of carvedilol in human liver and intestinal microsomes. Pharmacology. 2012;90 (3-4) :117-24.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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