Thiethylperazine-d3

CAT: 0804-HY-B1794SSize: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-B1794SSize:1 Each
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Description
Thiethylperazine-d3 is the deuterium labeled Thiethylperazinee (HY-B1794) . Thiethylperazine, a phenothiazine derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist. Thiethylperazine is also a selective ABCC1activator that reduces amyloid-β (Aβ) load in mice. Thiethylperazine has anti-emetic, antipsychotic and antimicrobial effects[1][2][3].
UNSPSC
12352005
Target
Amyloid-β; Bacterial; Dopamine Receptor; Histamine Receptor; Isotope-Labeled Compounds
Related Pathways
Anti-infection; GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling; Others
Field of Research
Infection; Neurological Disease
Smiles
CCSC(C=C1N2CCCN3CCN(C([2H])([2H])[2H])CC3)=CC=C1SC4=C2C=CC=C4
Molecular Formula
C22H26D3N3S2
Molecular Weight
402.63
References & Citations
[1]Czeizel AE, et al. Case-control study of teratogenic potential of thiethylperazine, an anti-emetic drug. BJOG. 2003 May;110 (5) :497-9. |[2]Krohn M, et al. Cerebral amyloid-β proteostasis is regulated by the membrane transport protein ABCC1 in mice. J Clin Invest. 2011 Oct;121 (10) :3924-31. |[3]Rahbar M, et al. Enhancement of vancomycin activity by phenothiazines against vancomycin-resistant Enterococcus faecium in vitro. Basic Clin Pharmacol Toxicol. 2010 Aug;107 (2) :676-9.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported

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