SSTR4 agonist 5

• Description:

  SSTR4 agonist 5 (Compound 5) is the orally active agonist for somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. SSTR4 agonist 5 exhibits good stability in human/rat liver microsomes. SSTR4 agonist 5 inhibits mechanical hyperalgesia in rat models[1].

• UNSPSC:

  12352005

• Target:

  Somatostatin Receptor

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling

• Field of Research:

  Neurological Disease

• Smiles:

  O=C (C1C2CNCC12C) NC (C) (C) C3=NC4=C5C (CCC4) =CC=CN35

• Molecular Formula:

  C20H26N4O

• Molecular Weight:

  338.45

• References & Citations:

  [1]Qiu G, et al., Nitrogen-containing heterocyclic compound, pharmaceutical composition, and applications. WO2022012534

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• Isoform:

  SSTR4

• CAS Number:

  2761347-44-6