SSTR4 agonist 5

• CAS Number :

  2761347-44-6

• Target :

  Somatostatin

• Related Pathways :

  GPCR/G Protein

• Bioactivity :

  SSTR4 agonist5 (Compound 5) is an orally active agonist of the somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. It demonstrates good stability in human/rat liver microsomes and can inhibit mechanical hyperalgesia in rat models.

• Smiles :

  O=C(NC(C1=NC2=C3C(=CC=CN13)CCC2)(C)C)C4C5CNCC45C

• Molecular Formula :

  C20H26N4O

• Molecular Weight :

  338.447

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C