SSTR4 agonist 5

• Target:

  Somatostatin

• Related Pathways:

  GPCR/G Protein

• Bioactivity:

  SSTR4 agonist5 (Compound 5) is an orally active agonist of the somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. It demonstrates good stability in human/rat liver microsomes and can inhibit mechanical hyperalgesia in rat models.

• Smiles:

  O=C (NC (C1=NC2=C3C (=CC=CN13) CCC2) (C) C) C4C5CNCC45C

• Molecular Formula:

  C20H26N4O

• Molecular Weight:

  338.447

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2761347-44-6