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3-Hydroxy darifenacin

CAT: 0804-HY-149504Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-149504Size:1 Each
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Description
3-Hydroxy darifenacin is a metabolite of Darifenacin. 3-Hydroxy darifenacin is an antagonist of M1-5 muscarinic receptors with Kis values of 17.78, 79.43, 2.24, 36.31 and 6.17 nM, respectively in CHO cells[1].
CAS Number
206048-82-0
UNSPSC
12352005
Hazard Statement
H302+H312+H332-H315-H319
Target
Drug Metabolite; mAChR
Related Pathways
GPCR/G Protein; Metabolic Enzyme/Protease; Neuronal Signaling
Field of Research
Neurological Disease
Smiles
NC(C(C1=CC=CC=C1)(C2=CC=CC=C2)[C@H]3CN(CC3)CCC4=CC=C(OCC5O)C5=C4)=O
Molecular Formula
C28H30N2O3
Molecular Weight
442.55
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P501
References & Citations
[1]Mansfield KJ, et al. Comparison of receptor binding characteristics of commonly used muscarinic antagonists in human bladder detrusor and mucosa. J Pharmacol Exp Ther. 2009 Mar;328 (3) :893-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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