DG013B (formate)

• Description :

  DG013B formate is an epimer of DG013A (HY-139907) . DG013B formate has weak affinity for ERAP1 and ERAP2 and is often used as a negative control to study the binding properties of DG013A and its analogues to ERAP1 and ERAP2[1].

• UNSPSC :

  12352005

• Target :

  Aminopeptidase

• Related Pathways :

  Metabolic Enzyme/Protease

• Field of Research :

  Others

• Purity :

  99.57

• Smiles :

  O=P([C@@H](N)CCC1=CC=CC=C1)(O)C[C@H](CC(C)C)C(N[C@H](C(N)=O)CC2=CNC3=CC=CC=C23)=O.O=CO.O=CO.O=CO

• Molecular Formula :

  C30H43N4O10P

• Molecular Weight :

  650.66

• References & Citations :

  [1]Birgit Wilding, et al. Investigating the phosphinic acid tripeptide mimetic DG013A as a tool compound inhibitor of the M1-aminopeptidase ERAP1. Bioorg Med Chem Lett. 2021 Jun 15;42:128050.

• Shipping Conditions :

  Blue Ice

• Storage Conditions :

  -20°C (Powder, sealed storage, away from moisture)

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported