PF-05212377
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


PF-05212377
Bioactivity:
PF-05212377 (SAM-760) is an inhibitor of the serotonin receptor 5-HT6. It acts as a substrate for the human transport proteins P-gp/non-BCRP. The compound has demonstrated blood-brain barrier permeability in non-human primates. PF-05212377 is utilized in research related to Alzheimers disease.Smiles:
O=S (=O) (C=1C=CC=CC1) N2C3=CC=CC (=C3N=C2C) N4CCNCC4Molecular Formula:
C18H20N4O2SMolecular Weight:
356.44Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
1226793-34-5
