Products for Research Use Only

Caloxin 1C2

CAT: 0931-T89159-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T89159-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Proton pump, Calcium Channel
Related Pathways
Membrane transporter/Ion channel, Metabolism
Bioactivity
Caloxin 1C2 is a specific inhibitor of PMCA (plasma membrane Ca2+-ATPases), displaying selective affinity for PMCA4 over PMCA1, 2, and 3. The Ki values for Caloxin 1C2 are 2.3 μM for PMCA4 and 21 μM for PMCA1. Notably, Caloxin 1C2 does not significantly affect overall Ca2+ transport. Additionally, it impacts the contractile force of coronary arteries.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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