A3AR agonist 4

• Target:

  Adenosine Receptor

• Related Pathways:

  GPCR/G Protein|||Neuroscience

• Bioactivity:

  A3AR agonist 4, an A3 adenosine receptor (A3AR) agonist, exhibits an inhibitory affinity (K i) of 1.24 nM for hA3AR and dampens cAMP production with an EC 50 value of 0.17 nM. It is utilized in the study of inflammation and pain [1].

• Smiles:

  O[C@@H]1[C@]2([C@](C2)([C@H]([C@@H]1O)N3C4=C(N=C3)C5=C(C(Cl)=N4)C=C(C)N5)[H])C6=NN(C)C=N6

• Molecular Formula:

  C18H18ClN7O2

• Molecular Weight:

  399.83

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  3032475-23-0