A3AR agonist 1

• Target:

  Adenosine Receptor

• Related Pathways:

  Neuroscience|||GPCR/G Protein

• Bioactivity:

  A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes ?-arrestin2 recruitment with an effective concentration (EC50) of 5.17 nM. It serves as a research tool in various pathological conditions, including inflammatory diseases, ischemia, cancer, neuropathic pain, and liver diseases [1].

• Molecular Formula:

  C28H34N6O6

• Molecular Weight:

  550.61

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C