PRMT4-IN-2

CAT:
931-T81399-01
Size:
5 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
PRMT4-IN-2 - image 1

PRMT4-IN-2

  • Target:

    Histone Methyltransferase|||Others
  • Related Pathways:

    Others|||Chromatin/Epigenetic
  • Bioactivity:

    PRMT4-IN-2 (compound 55) acts as a pan-inhibitor across various protein arginine methyltransferase (PRMT) isoforms, exhibiting inhibitory potencies with IC50 values of 92 nM for PRMT4, 436 nM for PRMT6, 460 nM for PRMT1, 823 nM for PRMT8, and 1.386 ?M for PRMT3 [1].
  • Shipping Conditions:

    Cool pack
  • Storage Temperature:

    -20°C