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DCLK1-IN-2

CAT: 0931-T79421-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T79421-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2978517-43-8
Target
Others, Serine Protease
Related Pathways
Others, Proteases/Proteasome
Bioactivity
DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cell lines with an IC50 of 0.6 μM, as well as in vivo antitumor potency [1].
Smiles
N(C1=C2C(=NC(NC3=C(OC)C=C(C=C3)N4CCN(C)CC4)=N1)N=CN2)C5=C(S(C(C)C)(=O)=O)C=CC=C5
Molecular Formula
C26H32N8O3S
Molecular Weight
536.65
Shipping Conditions
Ice Packs
Storage Temperature
-20°C