CBP-IN-1

• Target:

  Epigenetic Reader Domain

• Related Pathways:

  Chromatin/Epigenetic

• Bioactivity:

  CBP-IN-1 (compound 12) is a potent CBP inhibitor with an IC50 of 1.5 nM, additionally suppressing CBP BRET and BRD4 (1) with IC50 values of 690 nM and 3100 nM, respectively [1].

• Smiles:

  C(C)(=O)N1CC=2C(=NN(C2CC1)C3CCNCC3)N4C=5C(=CC(=C(C(F)F)C5)C6=CN(C)N=C6)CCC4

• Molecular Formula:

  C27H33F2N7O

• Molecular Weight:

  509.59

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1936431-44-5