Analgesic agent-2

• Target:

  Sodium Channel

• Related Pathways:

  Membrane transporter/Ion channel

• Bioactivity:

  Analgesic Agent-2, a selective orally active inhibitor of the NaV1.8 channel, demonstrates an IC50 of 50.18 nM in HEK293 cells that stably express the human NaV1.8 channel, indicating its potential for analgesic activity [1].

• Molecular Formula:

  C21H21ClF2N4O2

• Molecular Weight:

  434.87

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C